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Palosuran hydrochloride 540769-28-6(free base）
CAS No.
Palosuran hydrochloride 540769-28-6(free base） ( —— )
Catalog No. M17710 CAS No.
Palosuran is a new potent and specific antagonist of the human UT receptor with an IC50 of 3.6±0.2 nM.
Purity : 98%
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 188 | Get Quote |
|
| 10MG | 292 | Get Quote |
|
| 25MG | 474 | Get Quote |
|
| 50MG | 677 | Get Quote |
|
| 100MG | Get Quote | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NamePalosuran hydrochloride 540769-28-6(free base）
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NoteResearch use only, not for human use.
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Brief DescriptionPalosuran is a new potent and specific antagonist of the human UT receptor with an IC50 of 3.6±0.2 nM.
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DescriptionPalosuran is a new potent and specific antagonist of the human UT receptor with an IC50 of 3.6±0.2 nM.
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Synonyms——
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PathwayPI3K/Akt/mTOR signaling
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TargetPI3K
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RecptorUrotensin Receptor (GPR14)
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Research Area——
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Indication——
Chemical Information
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CAS Number--
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Formula Weight454.99
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Molecular FormulaC25H31ClN4O2
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Purity98%
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Solubility——
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SMILESCl.Cc2nc1ccccc1c(c2)NC(=O)NCCN3CCC(O)(CC3)Cc4ccccc4
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Clozel M, et al. J Pharmacol Exp Ther, 2004, 311(1):204-212.
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